Publicaciones 2016-2017

Nuevas publicaciones (+2018...) y más información en:

Efficient total synthesis of neocryptolepine and synthetic access to 6-methylquinindoline from a common intermediate. María V. Méndez, Daniel A. Heredia, Enrique L. Larghi, Andrea B. J. Bracca y Teodoro S. Kaufman. RSC Adv. 7, 28298-28307 (2017). RSC Adv 2017 7 28298.pdf

Convenient Michael Addition/b-elimination Approach to the Synthesis of 4-Benzyl- and 4-Aryl-selenyl Coumarins using Diselenides as Selenium Sources. Gustavo Padilha, Paloma T. Birmann, Micaela Domingues, Teodoro S. Kaufman, Lucielli Savegnago y Claudio C. Silveira. Tetrahedron Lett. 58, 985-990 (2017).

Synthesis of Chromeno[4,3-b]pyrrol-4(1H)-ones, from b-Nitroalkenes and 4-Phenylaminocoumarins, under Solventless Conditions. Gustavo Padilha, Bernardo A. Iglesias, Davi F. Back, Teodoro S. Kaufman y Claudio C. Silveira. ChemistrySelect 2, 1297-1304 (2017). ChemistrySelect 2017 2 1297.pdf

First Total Synthesis of the Only Known 2-Isopropyliden-2H-benzofuran-3-one Isolated from V. luetzelburgii", Jorgelina L. Pergomet, Enrique L. Larghi, Teodoro S. Kaufman y Andrea B. J. Bracca. RSC Adv. 7, 5242-5250 (2017). RSC Adv 2017 7 5242.pdf

A Computational Chemistry-Driven Solution to Rubriflordilactone B". Nicolás Grimblat, Teodoro S. Kaufman y Ariel M. Sarotti. Org. Lett. 18, 6420-6423 (2016). Org Lett 2016 18 6420.pdf

Determination of the Main Solid-State Form of Albendazole in Bulk Drug, Employing Raman Spectroscopy Coupled to Multivariate Analysis. Natalia L. Calvo, Aida Ben Altabef, Marcelo Arias, Rubén M. Maggio y Teodoro S. Kaufman. J. Pharm. Biomed. Anal. 129, 190-197 (2016).  J Pharm Biomed Anal 2016 129 190.pdf

The 3,4-Dioxygenated 5-Hydroxy-4-aryl-quinolin-2(1H)-one Alkaloids. Results of 20 Years of Research, Uncovering a New Family of Natural Products. Sebastian O. Simonetti, Enrique L. Larghi y Teodoro S. Kaufman. Nat. Prod. Rep. 33, 1425-1446 (2016). Nat Prod Rep 2016 33 1425.pdf
A Theoretical Study of the Duff Reaction: Insights into its Selectivity. Nicolás Grimblat, Ariel M. Sarotti, Teodoro S. Kaufman y Sebastian O. Simonetti. Org. Biomol. Chem. 14, 10496-10501 (2016). Org Biomol Chem 2016 14 10496.pdf
Wittig-Horner Mediated Synthesis of 4-Vinyl Sulfide Derivatives of Pyrazoles. Gustavo Padilha, Teodoro S. Kaufman y Claudio C. Silveira. Tetrahedron Lett. 57, 3349-3353 (2016). Tetrahedron Lett 2016 57 3349.pdf
Mebendazole Crystal Forms in Tablet Formulations. An ATR-FTIR/Chemometrics Approach to Polymorph Assignment. Natalia L. Calvo, Rubén M. Maggio y Teodoro S. Kaufman. J. Pharm. Biomed. Anal. 122, 157-165 (2016).  J Pharm Biomed Anal 2016 122 157.pdf
Expedient Approach to 6-Bromo-2-isopropylidenecoumaranone, a Potential Intermediate for the Synthesis of TMC-120B, Pseudodeflectusin and their Congeners. Jorgelina L. Pergomet, Teodoro S. Kaufman y Andrea B. J. Bracca. Helv. Chim. Acta 99, 398-404 (2016). Helv Chim Acta 2016 99 398.pdf
A Straightforward Synthesis of 5-Methylaaptamine from Eugenol, Employing a 6π-Electrocyclization Reaction of a 1-Azatriene. Daniel A. Heredia, Enrique L. Larghi y Teodoro S. Kaufman. Eur. J. Org. Chem. 1397-000 (2016). Eur J Org Chem 2016 1397-1404.pdf.
Convenient Approach to an Advanced Intermediate Toward the Naturally Occurring, Bioactive 6-Substituted 5-Hydroxy-4-aryl-1H-quinolin-2-ones. Sebastián O. Simonetti, Enrique L. Larghi y Teodoro S. Kaufman. Org. Biomol. Chem. 14, 2625-2636 (2016). Org Biomol Chem 2016 14 2625.pdf
Preparation and Physical Characterization of a Diclofenac-Ranitidine Co-precipitate for Improving the Dissolution of Diclofenac. Robertino O. Gaitano, Natalia L. Calvo, Griselda E. Narda, Teodoro S. Kaufman, Rubén M. Maggio y Elena V. Brusau. J. Pharm. Sci. 105, 1258-1268 (2016). J Pharm Sci 2016 105 1258.pdf
Synthesis and Preliminary Evaluation of 3-Thiocyanato-1H-indoles asPotential Anticancer Agents. Margiani P. Fortes, Paulo B. N. da Silva, Teresinha G. da Silva, Teodoro S. Kaufman, Gardenia C. G. Militao y Claudio C. Silveira. Eur. J. Med. Chem. 118, 21-26 (2016). Eur J Med Chem 2016 118 21.pdf